2. Signaling Pathways
  3. Metabolic Enzyme/Protease
  4. Drug Metabolite

Drug Metabolite

Drug Metabolite

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Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-W587742
    Dicyclohexylammonium 3-hydroxy-1-methylpropylmercapturic acid
    Dicyclohexylammonium 3-hydroxy-1-methylpropylmercapturic acid is a metabolite of Crotonaldehyde. Crotonaldehyde is an organic aldehyde, mainly used for the synthesis of plastics, drugs and fragrances, etc.
    Dicyclohexylammonium 3-hydroxy-1-methylpropylmercapturic acid
  • HY-135394R
    3-Desacetyl Cefotaxime lactone (Standard)
    3-Desacetyl Cefotaxime lactone (Standard) is the analytical standard of 3-Desacetyl Cefotaxime lactone. This product is intended for research and analytical applications. 3-Desacetyl Cefotaxime lactone is the active metabolite of Cefotaxime. Cefotaxime sodium salt is a third-generation cephalosporin antibiotic.
    3-Desacetyl Cefotaxime lactone (Standard)
  • HY-133694R
    2-Aminoflubendazole (Standard)
    2-Aminoflubendazole (Standard) is the analytical standard of 2-Aminoflubendazole. This product is intended for research and analytical applications. 2-Aminoflubendazole is the metabolite of Benzimidazoles. Benzimidazoles (BZ) are a class of agents with activities against fungi, protozoa, and helminthes.
    2-Aminoflubendazole (Standard)
  • HY-113095R
    γ-CEHC (Standard)
    Ftivazide (Standard) is the analytical standard of Ftivazide. This product is intended for research and analytical applications. Ftivazide has anti-tuberculosis activity.
    γ-CEHC (Standard)
  • HY-W016221R
    6-Hydroxy Chlorzoxazone (Standard)
    6-Hydroxy Chlorzoxazone (Standard) is the analytical standard of 6-Hydroxy Chlorzoxazone. This product is intended for research and analytical applications. 6-Hydroxy Chlorzoxazone is a metabolite of Chlorzoxazone (HY-B1462). Chlorzoxazone is a centrally acting muscle relaxant used to treat muscle spasm and the resulting pain or discomfort.
    6-Hydroxy Chlorzoxazone (Standard)
  • HY-126129R
    Desacetylcefotaxime (Standard)
    Desacetylcefotaxime (Standard) is the analytical standard of Desacetylcefotaxime. This product is intended for research and analytical applications. Desacetylcefotaxime, the in vivo metabolite of Cefotaxime (CTX), possesses significant in vitro antimicrobial activity similar to the parent compound against a variety of aerobic and anaerobic bacteria.
    Desacetylcefotaxime (Standard)
  • HY-N8483
    Eprinomectin B1a
    Eprinomectin B1a is a Eprinomectin (HY-12643) metabolite (an antiparasitic compound).
    Eprinomectin B1a
  • HY-G0001
    Lurasidone metabolite 14283
    Lurasidone metabolite 14283 is an active metabolite of lurasidone (HY-B0032A) and can be used in antipsychotic research.
    Lurasidone metabolite 14283
  • HY-172565
    Posaconazole D-glucuronide
    Posaconazole D-glucuronide (SCH 56592 D-glucuronide) is a glucuronide metabolite of the antifungal agent Posaconazole (HY-17373). Posaconazole D-glucuronide can be formed in human liver microsomes catalyzed by UGT1A4.
    Posaconazole D-glucuronide
  • HY-W750297
    p,p'-DDD-13C12
    p,p'-DDD-13C12 is 13C labeled p,p'-DDD. p,p'-DDD is a major metabolite of p,p'-DDT. p,p'-DDD occurs in the feces and livers of rats, that are given p,p'-DDT by stomach tube, but not of rats injected intraperitoneally with p,p'-DDT.
    p,p'-DDD-<sup>13</sup>C<sub>12</sub>
  • HY-W588198
    1,2-Cyclohexanedicarboxylic acid mono 4-methyl-7-carboxy-heptyl ester
    1,2-Cyclohexanedicarboxylic Acid Mono 4-Methyl-7-carboxy-heptyl Ester is a secondary oxidized metabolite of di(isononyl) cyclohexane-1,2-dicarboxylate (DINCH) , an alternative for phthalate plasticizer.
    1,2-Cyclohexanedicarboxylic acid mono 4-methyl-7-carboxy-heptyl ester
  • HY-W020576S
    Rivastigmine metabolite-d6
    Rivastigmine metabolite-d6 (NAP 226-90-d6) is a deuterated form of Rivastigmine metabolite. Rivastigmine metabolite (NAP 226-90) is a metabolite produced by the hydrolysis of Rivastigmine (HY-17368). Rivastigmine metabolite serves as a surrogate marker to track the bioavailability, metabolic extent, and transdermal patch delivery rate of Rivastigmine.
    Rivastigmine metabolite-d<sub>6</sub>
  • HY-125850R
    Berberrubine chloride (Standard)
    Berberrubine (chloride) (Standard) is the analytical standard of Berberrubine (chloride). This product is intended for research and analytical applications. Berberrubine chloride is an orally active metabolite of berberine. Berberrubine chloride alleviates mucosal lesions and inflammation in mouse colitis models. Berberrubine chloride has anti-inflammatory, anti-tumor, and antiviral activities.
    Berberrubine chloride (Standard)
  • HY-W410706
    1-Salicylate glucuronide
    1-Salicylate glucuronide is a metabolite of Salicylic acid (HY-B0167) and Aspirin (HY-14654).
    1-Salicylate glucuronide
  • HY-150159S
    Cotinine-d3 N-β-D-Glucuronide
    Cotinine-d3 N-β-D-Glucuronide is the deuterium labeled Cotinine N-β-D-Glucuronide (HY-W588194). Cotinine N-β-D-Glucuronide is a glucuronide conjugate of the tobacco metabolite Cotinine (HY-B1178). Cotinine N-β-D-Glucuronide is promising for research of tobacco carcinogen metabolism and cognitive function.
    Cotinine-d<sub>3</sub> N-β-D-Glucuronide
  • HY-185226
    γ-Linolenic acid NHS ester
    γ-Linolenic acid NHS ester is a lipid metabolite of γ-Linolenic acid (GLA) (HY-N7140), which can serve as a synthetic intermediate or probe labeling reagent for the preparation of GLA conjugates. In practical applications, γ-Linolenic acid NHS ester can be conjugated with taxanes and polysaccharides to form dual-type conjugates for drug delivery purposes.
    γ-Linolenic acid NHS ester
  • HY-W015169R
    5-Methoxytryptamine (Standard)
    5-Methoxytryptamine (Standard) is the analytical standard of 5-Methoxytryptamine (HY-W015169). This product is intended for research and analytical applications. 5-Methoxytryptamine, a metabolite of Melatonin, is a nonselective 5-HT receptor agonist. 5-Methoxytryptamine has no affinity for the 5-HT3 receptor. 5-Methoxytryptamine is also a potent antioxidant and has radioprotective action.
    5-Methoxytryptamine (Standard)
  • HY-15852
    THRX-195518
    THRX-195518 is the major metabolite of Revefenacin (HY-15851), a lung-selective and long-acting muscarinic antagonist. THRX-195518 can be utilized in research related to chronic obstructive pulmonary disease.
    THRX-195518
  • HY-W086896R
    α-Demethylnaproxen (Standard)
    α-Demethylnaproxen (Standard) is the analytical standard of α-Demethylnaproxen (HY-W086896). This product is intended for research and analytical applications. α-Demethylnaproxen (Compound 6-MNA) is the major metabolite of Nabumetone (HY-B0559). Nabumetone is an orally active non-acidic anti-inflammatory agent, acts as a potent and selective COX-2 inhibitor.
    α-Demethylnaproxen (Standard)
  • HY-G0012S
    Monohydroxy Netupitant-d6
    Monohydroxy Netupitant-d6 is the deuterium labeled Monohydroxy Netupitant, which is a metabolite of Netupitant.
    Monohydroxy Netupitant-d<sub>6</sub>
Cat. No. Product Name / Synonyms Application Reactivity